平安! 发表于 2011-11-9 19:57 2 M- V9 t* A8 Z/ J+ T; Y. D; p
Pazopanib (100 mg/kg/day free base equivalent) * a+ l( @- k& R9 G8 F
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。: H* ^" d3 `2 @5 G" ]
搜索了一下,原料一大堆。* Y7 J" g, Y6 ~' A
' M/ V) u+ \3 C7 {& Z- K4 d对不起!100mg/kg是用于移植瘤的,我弄错了。- _) G8 ?5 l' |: ~ ~8 E
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以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------
2 j4 r$ ?& ?5 k$ A+ w! t% k* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
7 M: C" z, o' Z4 b% ]7 p% B& o# p* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
" z7 p9 \/ U- y! \" H6 X" E---------------------DOSAGE FORMS AND STRENGTHS --------------
9 H3 f# }5 f. c# Z200 mg tablets. (3)
2 P5 `0 I7 B9 ]-------------------------------CONTRAINDICATIONS------------------------ |